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Therapeutics

From a scaffold to a calibrated clearance estimate.

The molecule-side funnel, end to end. Profile a series for ADMET and compliance, optimize the leads, dock against the target with strain correction, and gate on a calibrated Phase I clearance estimate. Every stage runs inside the assistant.

predict_admetdock_with_strainlead_optimizationpredict_clinical_outcomescheck_compliancerun_molecular_dynamics

Toxicity and drug-like properties drive roughly 40 to 45 percent of clinical failures. NovoMCP surfaces those flags in silico, before a dollar of lab spend.

One instruction

What it looks like in practice.

any MCP-compatible assistant
you Profile this scaffold for ADMET and compliance, then dock the clean candidates against EGFR.
resolved 4 analogs · ran batch_profile across 84 properties
flagged 1 hERG liability and 1 PAINS alert via check_compliance (FAVES)
docked 3 survivors with dock_with_strain · top pose −9.4 kcal/mol
gated on predict_clinical_outcomes · calibrated Phase I clearance 0.71
Benchmarked

The accuracy, stated plainly.

0.756
NovoExpert-3
Phase I AUROC
0.535
pKa v9
SAMPL7 RMSE
31
ML ADMET
models
3/22
TDC ADMET endpoints
beat the current #1

ADMET on every compound

Absorption, distribution, metabolism, excretion, and toxicity. 31 endpoints via the NovoExpert model family, called against any SMILES you give the engine. Runs locally, on demand, results returned immediately.

Docking with strain correction

AutoDock-GPU poses, corrected for internal ligand strain so the binding estimate survives a medicinal chemist's scrutiny. Reference-ligand co-docking keeps the pose honest.

Lead optimization that respects the series

Scaffold-aware, property-directed optimization. Tanimoto thresholds tuned to the 0.80–0.85 sweet spot so generated analogs stay synthesizable and on-series.

A clinical-outcome gate, calibrated

NovoExpert-3 estimates Phase I clearance from physicochemical, ADMET, and target/indication features. Strong on cardiovascular and GI. The engine states its validated scope on every response.

Research preview

Run the molecule-side funnel on an engine you can audit.

NovoMCP is open to a small group of PIs, postdocs, and research engineers. Tell us what you are working on.